1236699-92-5Pimasertib (AS-703026)

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商品编号：A125227

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商品名称：1236699-92-5Pimasertib (AS-703026)
商品毛重：0.00
单位：件
上架时间：2017-10-31 22:40:36

名称: Pimasertib (AS-703026)英文名称: Pimasertib (AS-703026)≥98%产品编号 A125227
CAS号: 1236699-92-5分子式 C₁₅H₁₅FIN₃O₃分子量431.20

属性

溶解性	DMSO ≥83mg/mL Water
存贮条件	储存温度-20°C

描述

产品介绍	Pimasertib (AS-703026) is a highly selective, potent, ATP non-competitive allosteric inhibitor of MEK1/2 with IC50 of 5 nM-2 μM in MM cell lines.
别名	MSC1936369B;AS703026;N-[(2S)-2,3-二羟基丙基]-3-[(2-氟-4-碘苯基)氨基]-4-吡啶甲酰胺;MSC1936369B;AS-703026;AS 703026;N-[(2S)-2,3-Dihydroxypropyl]-3-[(2-fluoro-4-iodophenyl)amino]-4-pyridinecarboxamide
生化机理	AS703026 is a highly selective and potent noncompetitive inhibitor of MEK1 and MEK2 (IC50 = 5-11 nM).
备注	AS-703026 is a highly selective, potent, ATP non-competitive allosteric inhibitor of MEK1/2 with IC50 of 5 nM-2 μM in MM cell lines. Phase 1/2.
应用	A potent inhibitor of MEK1 and MEK2.